BDBM50341148 (E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo[d]imidazol-1-yl)prop-1-enyl)phenoxy)propanoic acid::CHEMBL1760558

SMILES Cc1ccc(cc1)C(=O)c1nc2ccccc2n1C\C=C\c1cccc(OC(C)(C)C(O)=O)c1

InChI Key InChIKey=KMHNYIMVDBRUQH-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50341148   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341148((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo...)
Affinity DataEC50:  1.70E+3nMAssay Description:Partial agonist activity at human PPARgamma expressed in CHO cells co-transfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341148((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo...)
Affinity DataEC50:  1.70E+3nMAssay Description:Partial agonist activity at mouse PPARalpha expressed in CHO cells co-transfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50341148((E)-2-methyl-2-(3-(3-(2-(4-methylbenzoyl)-1H-benzo...)
Affinity DataEC50:  3.60E+3nMAssay Description:Partial agonist activity at human PPARalpha expressed in CHO cells co-transfected with Gal4-responsive luciferase reporter plasmid after 24 hrs by tr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed