BDBM50337996 1-(1-(cyclohexylmethyl)-6-methoxy-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea::CHEMBL1684269

SMILES COc1ccc2N(CC3CCCCC3)CCC(NC(=O)Nc3cccc4[nH]ncc34)c2c1

InChI Key InChIKey=XFXAXIXVJKIEKT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50337996   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50337996(1-(1-(cyclohexylmethyl)-6-methoxy-1,2,3,4-tetrahyd...)Copy SMILESCopy InChI

Affinity DataIC50: 196nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of calcium influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/24/2011
Entry Details Article
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