BDBM50337994 1-(1-benzyl-6-tert-butyl-1,2,3,4-tetrahydroquinolin-4-yl)-3-(1H-indazol-4-yl)urea::CHEMBL1684267

SMILES CC(C)(C)c1ccc2N(Cc3ccccc3)CCC(NC(=O)Nc3cccc4[nH]ncc34)c2c1

InChI Key InChIKey=SFXDORUIZFRXSG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50337994   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50337994(1-(1-benzyl-6-tert-butyl-1,2,3,4-tetrahydroquinoli...)Copy SMILESCopy InChI

Affinity DataIC50: 121nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of calcium influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/24/2011
Entry Details Article
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