BDBM50336157 4-bromo-5-(4-bromophenyl)-N-cyclopentylisoxazole-3-carboxamide::CHEMBL1669545

SMILES Brc1c(noc1-c1ccc(Br)cc1)C(=O)NC1CCCC1

InChI Key InChIKey=SHBGWSIPKFLWGC-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50336157   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharpe and Dohme

Curated by ChEMBL

LigandBDBM50336157(4-bromo-5-(4-bromophenyl)-N-cyclopentylisoxazole-3...)Copy SMILESCopy InChI

Affinity DataIC50: 410nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium influx by fluorimetric assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/23/2011
Entry Details Article
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