BDBM50333774 (E)-(2-Methyl-4-{1-[4-methyl-2-(4-trifluoromethylphenyl)-thiazol-5-ylmethoxyimino]-ethyl}-phenoxy)-acetic acid::CHEMBL1644299

SMILES C\C(=N/OCc1sc(nc1C)-c1ccc(cc1)C(F)(F)F)c1ccc(OCC(O)=O)c(C)c1

InChI Key InChIKey=ODUUUGYLEOEHRQ-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50333774   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50333774((E)-(2-Methyl-4-{1-[4-methyl-2-(4-trifluoromethylp...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPARgamma expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50333774((E)-(2-Methyl-4-{1-[4-methyl-2-(4-trifluoromethylp...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human PPARalpha expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50333774((E)-(2-Methyl-4-{1-[4-methyl-2-(4-trifluoromethylp...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARdelta expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed