BDBM50331703 2,4-dichloro-6-(trifluoromethyl)-5,6,7,8,9,10-hexahydrocyclohepta[b]indol-6-ol::CHEMBL1290632

SMILES OC1(CCCCc2c1[nH]c1c(Cl)cc(Cl)cc21)C(F)(F)F

InChI Key InChIKey=UYVPMSMQBOHCIJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50331703   

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331703(2,4-dichloro-6-(trifluoromethyl)-5,6,7,8,9,10-hexa...)
Affinity DataIC50: 600nMT: 2°CAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Radius Health

US Patent
LigandPNGBDBM50331703(2,4-dichloro-6-(trifluoromethyl)-5,6,7,8,9,10-hexa...)
Affinity DataIC50: 600nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed