BDBM50324865 CHEMBL1221497::naphthalene-2-sulfonic acid [3-(4-methyl-piperazin-1-yl)-phenyl]-amide

SMILES CN1CCN(CC1)c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1

InChI Key InChIKey=VAEXXTRBLCNPTN-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50324865   

Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 5.15E+3nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]LSD from human 5HT7 expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 1.62E+3nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50324865(naphthalene-2-sulfonic acid [3-(4-methyl-piperazin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHOKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed