BDBM50322989 CHEMBL1210083::N-(1-(3,5-diethoxy-4-(1H-imidazol-1-yl)benzyl)piperidin-4-yl)-5-methylnicotinamide

SMILES CCOc1cc(CN2CCC(CC2)NC(=O)c2cncc(C)c2)cc(OCC)c1-n1ccnc1

InChI Key InChIKey=YTYBDUVKLIFXAG-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50322989   

TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322989(N-(1-(3,5-diethoxy-4-(1H-imidazol-1-yl)benzyl)pipe...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322989(N-(1-(3,5-diethoxy-4-(1H-imidazol-1-yl)benzyl)pipe...)
Affinity DataKi:  11nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed