BDBM50321856 4-{2-[7-Hydroxy-5,6,7,8-tetrahydronaphthalen-1-ylamino]-5-[4-(trifluoromethyl)-phenyl]oxazol-4-yl}benzonitrile::CHEMBL1173690

SMILES OC1CCc2cccc(Nc3nc(c(o3)-c3ccc(cc3)C(F)(F)F)-c3ccc(cc3)C#N)c2C1

InChI Key InChIKey=KVUKMCYRADIGGS-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50321856   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50321856(4-{2-[7-Hydroxy-5,6,7,8-tetrahydronaphthalen-1-yla...)Copy SMILESCopy InChI

Affinity DataIC50: 2nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor expressed in human 1321 cells assessed as inhibition of capsaicin-induced in intracellular ca...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
12/31/2012
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