BDBM50321833 2-Methyl-8-{5-[4-(trifluoromethyl)phenyl]oxazol-2-ylamino}-1,2,3,4-tetrahydronaphthalen-2-ol::CHEMBL1173458

SMILES CC1(O)CCc2cccc(Nc3ncc(o3)-c3ccc(cc3)C(F)(F)F)c2C1

InChI Key InChIKey=DBTUSIKSRJSFQQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50321833   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50321833(2-Methyl-8-{5-[4-(trifluoromethyl)phenyl]oxazol-2-...)Copy SMILESCopy InChI

Affinity DataIC50: 840nMAssay Description:Antagonist activity at human recombinant TRPV1 receptor expressed in human 1321 cells assessed as inhibition of capsaicin-induced in intracellular ca...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
12/31/2012
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL