BDBM50311793 4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)biphenyl-3-carboxylic acid::CHEMBL1080470

SMILES CCCCOc1ccc(cc1CNC(=O)c1ccc(cc1F)C(F)(F)F)-c1cccc(c1)C(O)=O

InChI Key InChIKey=HCGPTXKJCXPTFR-UHFFFAOYSA-N

Data  7 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50311793   

TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Agonist activity at PPARalpha receptor expressed in HEK293 cells co-transfected with GAL4 by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at PPARdelta receptor expressed in HEK293 cells co-transfected with GAL4 by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  29nMAssay Description:Partial agonist activity at human recombinant PPARdelta LBD expressed in HEK293 cells co-transfected with Gal4 assessed as beta-galactosidase activit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Partial agonist activity at human recombinant PPARalpha LBD expressed in HEK293 cells co-transfected with Gal4 assessed as beta-galactosidase activit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  29nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  1.70E+5nMAssay Description:Partial agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed