BDBM50303572 CHEMBL571999::[1-((Tetrahydro-2H-pyran-4-yl)methyl](3-noradamantane)methanone

SMILES O=C(c1cn(CC2CCOCC2)c2ccccc12)C12CC3CC1CC(C2)C3

InChI Key InChIKey=WBROYFRREDXBEY-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50303572   

TargetCannabinoid receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303572([1-((Tetrahydro-2H-pyran-4-yl)methyl](3-noradamant...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303572([1-((Tetrahydro-2H-pyran-4-yl)methyl](3-noradamant...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303572([1-((Tetrahydro-2H-pyran-4-yl)methyl](3-noradamant...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed