BDBM50303569 (1-(2-Aminoethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)-methanone::CHEMBL576485

SMILES CC1(C)C(C(=O)c2cn(CCN)c3ccccc23)C1(C)C

InChI Key InChIKey=QKJAICLUPJKFRV-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50303569   

TargetCannabinoid receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303569((1-(2-Aminoethyl)-1H-indol-3-yl)(2,2,3,3-tetrameth...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303569((1-(2-Aminoethyl)-1H-indol-3-yl)(2,2,3,3-tetrameth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303569((1-(2-Aminoethyl)-1H-indol-3-yl)(2,2,3,3-tetrameth...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed