BDBM50302517 4-(1,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicotinonitrile::CHEMBL585681

SMILES Cc1c(Nc2c(\C=C\c3ccccc3)cncc2C#N)ccc2n(C)ccc12

InChI Key InChIKey=OLHUPCIDRDIHRN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50302517   

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302517(4-(1,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302517(4-(1,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed