BDBM50299839 3-(3-(1H-Imidazol-1-yl)propyl)-2,3-dihydro-7-methyl-2-thioxothieno[3,2-d]pyrimidin-4(1H)-one::CHEMBL565694

SMILES Cc1csc2CN(CCCn3ccnc3)C(=S)Nc12

InChI Key InChIKey=PHEYUECIVOQIOV-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50299839   

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299839(3-(3-(1H-Imidazol-1-yl)propyl)-2,3-dihydro-7-methy...)
Affinity DataKi:  360nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed