BDBM50298968 (1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)sulfonyl]-N-[4-(propan-2-yloxy)phenyl]-2-azabicyclo[2.2.2]octane-6-carboxamide::CHEMBL578249

SMILES CC(C)Oc1ccc(NC(=O)[C@@H]2C[C@@H]3CC[C@@H]2N(C3)S(=O)(=O)c2cn(C)cn2)cc1

InChI Key

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50298968   

TargetElongation of very long chain fatty acids protein 6(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 6(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 220nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 6(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 220nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL5 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 6(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 73nMAssay Description:Inhibition of C-terminal V5-epitope-tagged mouse ELOVL6 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 717nMAssay Description:Inhibition of C-terminal V5-epitope-tagged mouse ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed