BDBM50295940 2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine::CHEMBL562384

SMILES Cc1nc2cc(C)nc(C)n2c1CN1CCN(CC1)c1ccccn1

InChI Key InChIKey=URKAJHJBVOPDPZ-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50295940   

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander-Universit£T

Curated by ChEMBL
LigandPNGBDBM50295940(2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl...)
Affinity DataKi:  640nMAssay Description:Displacement of [3H]spiroperidol from human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander-Universit£T

Curated by ChEMBL
LigandPNGBDBM50295940(2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]spiroperidol from human cloned dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander-Universit£T

Curated by ChEMBL
LigandPNGBDBM50295940(2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Bovine)
Friedrich-Alexander-Universit£T

Curated by ChEMBL
LigandPNGBDBM50295940(2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [3H]SCH23390 from bovine dopamine D1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed