BDBM50293928 (R)-5-Chloro-1-(1-cyclopropylethyl)-3-(2,4,6-trimethylphenylamino)pyrazin-2(1H)-one::(R)-5-chloro-1-(1-cyclopropylethyl)-3-(mesitylamino)pyrazin-2(1H)-one::CHEMBL558280

SMILES C[C@H](C1CC1)n1cc(Cl)nc(Nc2c(C)cc(C)cc2C)c1=O

InChI Key InChIKey=NRCBXZPRZSUGCI-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50293928   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293928((R)-5-chloro-1-(1-cyclopropylethyl)-3-(mesitylamin...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293928((R)-5-chloro-1-(1-cyclopropylethyl)-3-(mesitylamin...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293928((R)-5-chloro-1-(1-cyclopropylethyl)-3-(mesitylamin...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]ovine-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed