BDBM50293484 (R)-4-((1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)methyl)-N-(1-(4-methoxyphenyl)ethyl)benzamide::CHEMBL562016

SMILES COc1ccc(cc1)[C@@H](C)NC(=O)c1ccc(CC2CCN(Cc3ccc4OCOc4c3)CC2)cc1

InChI Key InChIKey=XGHQCOKQRQZBOU-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50293484   

TargetMelanin-concentrating hormone receptor 1(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50293484((R)-4-((1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidi...)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at MCHR1 (unknown origin) expressed in CHO cells co-expressing aequorin incubated for 10 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50293484((R)-4-((1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidi...)
Affinity DataKi:  776nMAssay Description:Binding affinity to MCH1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed