BDBM50289422 CHEMBL26314::{3-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]-phenyl}-methanol

SMILES N[C@@H](CS)CNc1ccc(Oc2cccc(CO)c2)cc1

InChI Key InChIKey=JLEHTMFTKRDAEM-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50289422   

LigandPNGBDBM50289422({3-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy...)
Affinity DataIC50: 335nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 n...More data for this Ligand-Target Pair
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Date in BDB:
8/21/2010
Entry Details Article