BDBM50281705 1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea::CHEMBL169953

SMILES Clc1ccc(NC(=O)Nc2cc3c(c[nH]2)nc2ccccc32)cc1

InChI Key InChIKey=GQGZOEJMQCPFFD-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50281705   

LigandPNGBDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 85nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article