BDBM50275158 4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}butyric acid::CHEMBL515995

SMILES OC(=O)CCCc1ccc(OCCN(c2nccs2)c2ccccc2)cc1

InChI Key InChIKey=PCKMEEZOBNUBRO-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50275158   

TargetFree fatty acid receptor 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR120-G-alpha-16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed