BDBM50275075 CHEMBL4129832

SMILES OC(=O)CNC(=O)c1ncc(cc1O)-c1cn(Cc2cc(Cl)cc(Cl)c2)nn1

InChI Key InChIKey=NTLPKYOEAZYLGC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50275075   

TargetEgl nine homolog 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275075(CHEMBL4129832)
Affinity DataIC50: 231nMAssay Description:Inhibition of HIF-PHD2 (181 to 426 residues) (unknown origin) using FITC-HIF1-alpha (556 to 574 residues) as substrate after 60 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed