BDBM50274786 1-(3-bromo-4-methylphenyl)-N-isopropyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide::CHEMBL511368

SMILES CC(C)NC(=O)c1cn(-c2ccc(C)c(Br)c2)c2ncccc2c1=O

InChI Key InChIKey=PUJMTYXKBMSBRR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50274786   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Merck Frosst Center For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50274786(1-(3-bromo-4-methylphenyl)-N-isopropyl-4-oxo-1,4-d...)
Affinity DataIC50: 66.5nMAssay Description:Intrinsic inhibition of GST-fused human PDE4A expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed