BDBM50273519 CHEMBL4129930

SMILES CC1(C)N(Cc2c1cccc2C(N)=O)c1cnc(cn1)C(F)(F)F

InChI Key InChIKey=WTZJBEDUYUCGGN-UHFFFAOYSA-N

Data  12 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 12 hits for monomerid = 50273519   

TargetHistone deacetylase 1(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC1 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC7 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC2 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC5 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC8 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of NanoLuc-tagged HDAC11 (unknown origin) by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC11 expressed in baculoviral expression system using FAM-RHKK as substrate by electrophoretic mobility...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC3 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC4 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC9 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC10 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Forma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50273519(CHEMBL4129930)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length recombinant human HDAC6 using fluorescent-labeled peptide as substrate by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed