BDBM50272549 CHEMBL4125928

SMILES C[C@@H](NC(=O)NCc1ccc(cc1)C(C)(C)C)c1ccc(NS(C)(=O)=O)cc1

InChI Key InChIKey=YKLPUVUAAJRISU-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50272549   

TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272549(CHEMBL4125928)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272549(CHEMBL4125928)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed