BDBM50272512 CHEMBL4129792

SMILES Clc1cc(Cl)cc(Oc2ncc(cc2Cl)-c2nnc([nH]2)S(=O)(=O)CC2CC2)c1

InChI Key InChIKey=LTLPRWXMBOBTPL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50272512   

LigandPNGBDBM50272512(CHEMBL4129792)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human Nav1.7 expressed in HEK cells clamped to holding potential yielding 20 to 50% inactivation assessed as reduction in peak sodium c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed