BDBM50272039 CHEMBL4129773

SMILES Cc1ccc(Oc2ccc(CN3CCC(O)=C(C(=O)NCC([O-])=O)C3=O)nc2)cc1

InChI Key InChIKey=PORDUXDTGYPVDE-UHFFFAOYSA-M

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50272039   

TargetEgl nine homolog 1(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272039(CHEMBL4129773)
Affinity DataIC50: 69nMAssay Description:Inhibition of human PHD2 using FITC-HIF1-alpha as substrate after 10 mins in presence of 2-oxoglutarate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed