BDBM50271439 CHEMBL453689::Tyr-Pro-Phe-Phe-NHCH3

SMILES CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1

InChI Key InChIKey=WEITVBLLGNOHNQ-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50271439   

TargetDelta-type opioid receptor(Mouse)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50271439(Tyr-Pro-Phe-Phe-NHCH3 | CHEMBL453689)
Affinity DataIC50: 54.6nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50271439(Tyr-Pro-Phe-Phe-NHCH3 | CHEMBL453689)
Affinity DataIC50: 136nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50271439(Tyr-Pro-Phe-Phe-NHCH3 | CHEMBL453689)
Affinity DataKi:  29.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50271439(Tyr-Pro-Phe-Phe-NHCH3 | CHEMBL453689)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed