BDBM50269131 CHEMBL4073701

SMILES C[C@H]1CN(C[C@@H](C)O1)c1c(NC(=O)c2cccc(c2)-c2ccccn2)cccc1C(F)(F)F

InChI Key InChIKey=KHTDNEVIFXQOKO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50269131   

LigandPNGBDBM50269131(CHEMBL4073701)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of slow inactivated human NaV1.7 expressed in HEK293 cells at -20 mV holding potential after 5 mins by IonWorks electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2020
Entry Details Article
PubMed