BDBM50268749 CHEMBL4097005

SMILES O=C(COc1ccc2OCOc2c1)N(Cc1cccs1)c1ccn[nH]1

InChI Key InChIKey=DMRQUYUWMPGIJT-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50268749   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Senomyx

Curated by ChEMBL

LigandBDBM50268749(CHEMBL4097005)Copy SMILESCopy InChI

Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium level after 15 mins by Fluo-3-AM dye-based fl...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/6/2020
Entry Details Article
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