BDBM50268219 CHEMBL4073378

SMILES CCOc1cc(CN2CC3(C2)CC(=NO3)N2CCC(CC)(CC2)C(O)=O)cc(OCC)c1-c1ccc(F)cc1

InChI Key InChIKey=SKQRLFRQQOYFLV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50268219   

TargetSomatostatin receptor type 5(Mouse)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268219(CHEMBL4073378)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268219(CHEMBL4073378)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2020
Entry Details Article
PubMed