BDBM50265765 5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(2-{(S)-1-carboxy-3-[(2,4-dicarboxy-butyl)-hydroxy-phosphinoyl]-propylcarbamoyl}-ethyl)-adamantan-1-yl]-propionylamino}-3-carboxy-propyl)-hydroxy-phosphinoyl]-4-carboxy-pentanoic acid::CHEMBL508430

SMILES CC(C)(C)OC(=O)NC12CC3(CCC(=O)N[C@@H](CCP(O)(=O)CC(CCC(O)=O)C(O)=O)C(O)=O)CC(CCC(=O)N[C@@H](CCP(O)(=O)CC(CCC(O)=O)C(O)=O)C(O)=O)(CC(CCC(=O)N[C@@H](CCP(O)(=O)CC(CCC(O)=O)C(O)=O)C(O)=O)(C3)C1)C2

InChI Key

Data  5 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50265765   

TargetGlutamate carboxypeptidase 2(Human)
Justus-Liebig-Universitat Giessen

Curated by ChEMBL
LigandPNGBDBM50265765(5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(...)
Affinity DataKd:  0.800nMAssay Description:Binding affinity to PSMA in human LNCaP cells assessed as cell surface binding in phosphate-buffered saline bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Justus-Liebig-Universitat Giessen

Curated by ChEMBL
LigandPNGBDBM50265765(5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to PSMA in human PC3 cells assessed as cell surface binding in Tris-buffered saline bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Justus-Liebig-Universitat Giessen

Curated by ChEMBL
LigandPNGBDBM50265765(5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to PSMA in human PC3 cells assessed as cell surface binding in phosphate-buffered saline bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Justus-Liebig-Universitat Giessen

Curated by ChEMBL
LigandPNGBDBM50265765(5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(...)
Affinity DataKd:  0.600nMAssay Description:Binding affinity to PSMA in human PC3 cells assessed as cell surface binding in presence of 100% calf serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Justus-Liebig-Universitat Giessen

Curated by ChEMBL
LigandPNGBDBM50265765(5-[((S)-3-{3-[5-tert-Butoxycarbonylamino-3,7-bis-(...)
Affinity DataKd:  0.600nMAssay Description:Binding affinity to PSMA in human LNCaP cells assessed as cell surface binding in Tris-buffered saline bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed