BDBM50263952 4-(3-chlorophenyl)-N-methyl-N-(2-(piperidin-1-yl)ethyl)piperazine-1-carboxamide::CHEMBL489590

SMILES CN(CCN1CCCCC1)C(=O)N1CCN(CC1)c1cccc(Cl)c1

InChI Key InChIKey=RWKPIEGRBPYNIV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50263952   

TargetHistamine H3 receptor(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50263952(4-(3-chlorophenyl)-N-methyl-N-(2-(piperidin-1-yl)e...)
Affinity DataIC50: 297nMAssay Description:Inverse agonist activity at human cloned histamine H3 receptor assessed as inhibition of (R)-alpha-methylhistamine-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed