BDBM50263096 CHEMBL477181::N-cyclohexyl-6-(1-isopropylpiperidin-4-yloxy)-2-naphthamide

SMILES CC(C)N1CCC(CC1)Oc1ccc2cc(ccc2c1)C(=O)NC1CCCCC1

InChI Key InChIKey=CUPKCDUMNJWBHZ-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50263096   

TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(N-cyclohexyl-6-(1-isopropylpiperidin-4-yloxy)-2-na...)
Affinity DataEC50:  21nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(N-cyclohexyl-6-(1-isopropylpiperidin-4-yloxy)-2-na...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed