BDBM50262224 6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-6,7-dihydrothiazolo[5,4-c]pyridin-4(5H)-one::6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-benzo[b][1,4]oxazin-4(3H)-yl)-6,7-dihydrothiazolo[5,4-c]pyridin-4(5H)-one::CHEMBL512440

SMILES Cn1cc(cn1)-c1ccc2OCCN(c3nc4CC(C)(C)NC(=O)c4s3)c2c1

InChI Key InChIKey=WGINENHXAFXAQX-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50262224   

LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 32nMAssay Description:Inhibition of PI3K deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 78nMAssay Description:Inhibition of PI3K gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 295nMAssay Description:Inhibition of PI3K alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 540nMAssay Description:Inhibition of PI3K betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 32nMAssay Description:Inhibition of PI3KdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262224(6,6-dimethyl-2-(6-(1-methyl-1H-pyrazol-4-yl)-2H-be...)
Affinity DataIC50: 78nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed