BDBM50261961 (1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phenyl)methanone::CHEMBL469172

SMILES O=C(c1n[nH]c2ccccc12)c1ccccc1NCc1ccc2ncccc2c1

InChI Key InChIKey=HBSXWFBLJONDCO-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50261961   

TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 230nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 300nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50: 130nMAssay Description:Inhibition of KDR autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed