BDBM50261027 4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide::CHEMBL493816

SMILES COc1ccc(cc1)S(=O)(=O)NCCCN1CCN(CC1)c1ccc(F)cc1

InChI Key InChIKey=ZHZAXFCAXCANQE-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50261027   

Target5-hydroxytryptamine receptor 7(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50261027(4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]...)
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50261027(4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]...)
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50261027(4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50261027(4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]...)
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50261027(4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]...)
Affinity DataIC50: 4.89E+3nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed