BDBM50260953 CHEMBL4072044

SMILES Cc1c(c[nH]c1C(N)=O)-c1ccnc(C)c1

InChI Key InChIKey=GBEUJGXZRJILPH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50260953   

TargetCyclin-C/Cyclin-dependent kinase 8(Human)
Roche Innovation Center Shanghai

Curated by ChEMBL
LigandPNGBDBM50260953(CHEMBL4072044)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed