BDBM50257262 CHEMBL4093499

SMILES FC(F)(F)c1ccc(CNC(=O)c2cccc(CN3CCCCC3)c2)cc1

InChI Key InChIKey=DZKGORBEITZGMV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50257262   

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Rat)
Oklahoma Medical Research Foundation

Curated by ChEMBL
LigandPNGBDBM50257262(CHEMBL4093499)
Affinity DataIC50: 37nMAssay Description:Inhibition of PERK activation in rat INS-1 cells assessed as suppression of tunicamycin-induced CHOP mRNA expression after 8 hrs by qRT-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2019
Entry Details Article
PubMed