BDBM50255347 CHEMBL4081842

SMILES COc1cc(cc(c1O)[N+]([O-])=O)[C@@H](O)P(O)(=O)CC[C@H](N)C(O)=O

InChI Key InChIKey=PEXVMHLARUAHNC-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50255347   

TargetMetabotropic glutamate receptor 4(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255347(CHEMBL4081842)
Affinity DataEC50:  720nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2019
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 8(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255347(CHEMBL4081842)
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2019
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 6(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255347(CHEMBL4081842)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2019
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 7(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255347(CHEMBL4081842)
Affinity DataEC50:  6.30E+4nMAssay Description:Agonist activity at mGlu7 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2019
Entry Details Article
PubMed