BDBM50254924 CHEMBL465923::N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-methyl-1H-benzo[d]imidazol-2-ylthio)-1H-indol-4-yloxy)acetamide

SMILES Cn1c(Sc2c[nH]c3cccc(OCC(=O)NS(=O)(=O)c4cc(Cl)c(Cl)s4)c23)nc2ccccc12

InChI Key InChIKey=YJHQZSSSVNHKBJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50254924   

TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50254924(N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-meth...)
Affinity DataIC50: 10.5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50254924(N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-meth...)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed