BDBM50254070 2-(2-chloro-4-methoxyphenylsulfonyl)-2-methyl-N-(quinolin-3-yl)propanamide::CHEMBL466390

SMILES COc1ccc(c(Cl)c1)S(=O)(=O)C(C)(C)C(=O)Nc1cnc2ccccc2c1

InChI Key InChIKey=RAEOAJBOVOPUDI-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50254070   

TargetCannabinoid receptor 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50254070(2-(2-chloro-4-methoxyphenylsulfonyl)-2-methyl-N-(q...)
Affinity DataEC50:  148nMAssay Description:Agonist activity at human CB2 receptor expressed in SF9 cells assessed as inhibition of CP-55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50254070(2-(2-chloro-4-methoxyphenylsulfonyl)-2-methyl-N-(q...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CB1 receptor expressed in SF9 cells assessed as inhibition of CP-55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed