BDBM50253977 1-(1-methyl-3-(piperidin-1-ylsulfonyl)-1H-pyrazol-5-yl)-3-phenylurea::CHEMBL462694

SMILES Cn1nc(cc1NC(=O)Nc1ccccc1)S(=O)(=O)N1CCCCC1

InChI Key InChIKey=YTGOQZGHNWFRQP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50253977   

TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50253977(1-(1-methyl-3-(piperidin-1-ylsulfonyl)-1H-pyrazol-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50253977(1-(1-methyl-3-(piperidin-1-ylsulfonyl)-1H-pyrazol-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of endothelial lipaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed