BDBM50253976 1-(1,2-dimethyl-5-(piperidin-1-ylsulfonyl)-1H-pyrrol-3-yl)-3-phenylurea::CHEMBL518672

SMILES Cc1c(NC(=O)Nc2ccccc2)cc(n1C)S(=O)(=O)N1CCCCC1

InChI Key InChIKey=RJMOQFZPDXQREC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50253976   

TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50253976(1-(1,2-dimethyl-5-(piperidin-1-ylsulfonyl)-1H-pyrr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50253976(1-(1,2-dimethyl-5-(piperidin-1-ylsulfonyl)-1H-pyrr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of endothelial lipaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed