BDBM50251830 (Z)-2-(4-(methylsulfonyl)phenyl)-N-(thiazol-2-yl)-3-(thiophen-2-yl)acrylamide::CHEMBL516458

SMILES CS(=O)(=O)c1ccc(cc1)C(=C/c1cccs1)\C(=O)Nc1nccs1

InChI Key InChIKey=ZCRHVAOVNFNLDX-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50251830   

TargetHexokinase-4(Human)
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251830((Z)-2-(4-(methylsulfonyl)phenyl)-N-(thiazol-2-yl)-...)
Affinity DataEC50:  560nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed