BDBM50251029 (R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine dihydrochloride::CHEMBL458587

SMILES CN(C)c1ccc(cc1)-c1cc2CCN(C)[C@@H]3Cc4ccc(O)c(O)c4-c(c1)c23

InChI Key InChIKey=BSBMMXOBOAVGQD-UHFFFAOYSA-N

Data  3 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50251029   

TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataIC50: 484nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251029((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed