BDBM50247584 2-(2-Pyridyl)-isothiazol-3(2H)-one::CHEMBL489494

SMILES O=c1ccsn1-c1ccccn1

InChI Key InChIKey=LDQGZDZYAMGIRK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50247584   

TargetHistone acetyltransferase KAT2B(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50247584(2-(2-Pyridyl)-isothiazol-3(2H)-one | CHEMBL489494)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of GST-fused recombinant HAT PCAF expressed in Escherichia coli by filter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50247584(2-(2-Pyridyl)-isothiazol-3(2H)-one | CHEMBL489494)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of GST-fused recombinant HAT p300 expressed in Escherichia coli by filter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed