BDBM50240247 CHEMBL4095834

SMILES Fc1cc(OCC2NCCC=C2c2cccc(Cl)c2)c(Cl)cc1S(=O)(=O)Nc1cscn1

InChI Key InChIKey=PBWFMCSGENTSLG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50240247   

TargetSodium channel protein type 9 subunit alpha(Human)
Wuxi Apptec (Shanghai)

Curated by ChEMBL
LigandPNGBDBM50240247(CHEMBL4095834)
Affinity DataIC50: 580nMAssay Description:Inhibition of human Nav1.7 expressed in CHO-K1 cells at -120 mV holding potential incubated over 5 mins measured at 15 secs interval by Qpatch clamp ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2019
Entry Details Article
PubMed