BDBM50240207 CHEMBL4072863

SMILES CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(NCc4cccc(c4)-c4cccs4)c3)cc2C(F)(F)F)CC1

InChI Key InChIKey=LIBCJKPMHVGRLL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50240207   

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50240207(CHEMBL4072863)
Affinity DataIC50: 350nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2019
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50240207(CHEMBL4072863)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human c-Kit using poly[Glu:Tyr] (4:1) as substrate measured after 2 hrs in presence of [33gammaP]ATP by P18 ion exchange chromatographi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2019
Entry Details Article
PubMed